PROTAC 分子
提供PROTAC藥物開發所需關鍵材料,包括E3 ligase ligands、pre-assembled linker-ligase modules、linker building blocks與相關warhead結構。可協助研究者快速組裝PROTAC分子並進行結構活性關係研究。
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| Core → Functional group↓ |
Pomalidomide | Lenalidomide | VHL |
| Hydroxyl group (-OH) | 44 products | 54 products | na |
| Amine (-NH2) | 47 products | 41 products | 1 product |
| Nboc | 5 products | na | 4 products |
| Aldehyde | 1 product | na | na |
| Carboxylic acids | 6 products | 8 products | 1 product |
| Tert-butyl ester | 4 products | na | na |
| Bromine (-Br) | na | 1 products | na |
| Total quantity | 107 products | 104 products | 6 products |
| Download | PDF file | PDF file | PDF file |



